| Weight | 379.501 g/mol |
|---|---|
| Formula | C20H33N3O4 |
| Hydrogen Acceptors | 5 |
| Hydrogen Donors | 3 |
| Aromatic Rings | 1 |
| Rotatable Bonds | 9 |
celiprolol (56980-93-9)
Selectol · Celiprolol, Monohydrochloride, (R)-Isomer · Celiprolol Monohydrochloride
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- Transport of celiprolol across human intestinal epithelial (Caco-2) cells: mediation of secretion by multiple transporters including P-glycoprotein (British Journal of Pharmacology, 1993)
- Effect of celiprolol on prevention of cardiovascular events in vascular Ehlers-Danlos syndrome: a prospective randomised, open, blinded-endpoints trial (The Lancet, 2010)
- Itraconazole increases but grapefruit juice greatly decreases plasma concentrations of celiprolol. (Clinical Pharmacology & Therapeutics, 2003)
- Alterations in nitric oxide synthase activity, superoxide anion generation, and platelet aggregation in systemic hypertension, and effects of celiprolol. (American Journal of Cardiology, 1994)
- Impact of Curcumin-Induced Changes in P-Glycoprotein and CYP3A Expression on the Pharmacokinetics of Peroral Celiprolol and Midazolam in Rats (Drug Metabolism and Disposition, 2006)
- Orange juice substantially reduces the bioavailability of the adrenergicblocking agent celiprolol (Clinical Pharmacology & Therapeutics, 2004)
-
Predict GHS Hazards for Any Chemical in silico.
Including Acute Oral Tox, Skin Sensitization, Eye Irritation, Aquatic Tox, & more. - Selectol
- Celiprolol, Monohydrochloride, (R)-Isomer
- Celiprolol Monohydrochloride
- Celiprolol, (+,-)-Isomer
- Celiprolol, (R)-Isomer
- Celiprolol, (S)-Isomer
- REV5320A
- ST1396
- Celiprolol, Monohydrochloride, (S)-Isomer
- Celiprolol Hydrochloride
- N'-(3-Acetyl-4-(3-((1,1-dimethylethyl)amino)-2-hydroxypropoxy)phenyl)-N,N-diethylurea
- ST-1396
- REV 5320A
- REV-5320A
- ST 1396
-
SMILESCCN(CC)C(=O)NC1=CC(=C(C=C1)OCC(CNC(C)(C)C)O)C(=O)C
-
InChIKeyJOATXPAWOHTVSZ-UHFFFAOYSA-N
- Pubchem - celiprolol
- Wikipedia - celiprolol
Celiprolol (brand names Cardem, Selectol, Celipres, Celipro, Celol, Cordiax, Dilanorm) is a medication in the class of beta blockers, used in the treatment of high blood pressure. It has a unique pharmacology: it is a selective 1 receptor antagonist, but a 2 receptor partial agonist. It is also a weak 2 receptor antagonist.
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Synthesis
3-(3-Acetyl-4-hydroxyphenyl)-1,1-diethylurea
+
1-(tert-butylamino)-3-chloropropan-2-ol
(Williamson ether)
Reactant
+
DIETHYLAMINE
(Schotten-Baumann amide from acid)
tert-Butylamine
+
Reactant
(Alkylation of primary amines)
Reactant
+
ACETYL CHLORIDE
(Friedel-Crafts acylation)
Reactant
+
DIETHYLAMINE
(Thiourea)
Reactant
+
dimethyl sulfide
(Corey-Kim oxidation of secondary alcohols)
Acetonitrile
+
Reactant
(Grignard carbonyl)
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